Final API | Chemical Name | Cas no |
Sacubitril Valsartan | (R,E)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)aMino)-2-Methylpent -2-enoic acid | 1012341-48-8 |
(2R,4S)-5-(Biphenyl-4-yl)-4-[(tert-butoxycarbonyl)amino]-2-methylpentanoic acid | 1012341-50-2 | |
(2R,4S)-4-Amino-5-(biphenyl-4-yl)-2-methylpentanoic acid ethyl ester hydrochloride | 149690-12-0 | |
Sacubitril Calcium | 1369773-39-6 | |
Sacubitril Sodium | 149690-05-1 | |
Finerenone | 2-Cyanoethyl 4-(4-cyano-2-methoxyphenyl)-1,4,5,6-tetrahydro-2,8-dimethyl-5-oxo-1,6-naphthyridine-3-carboxylate | 1050477-43-4 |
2-Cyanoethyl 4-(4-cyano-2-methoxyphenyl)-5-ethoxy-1,4-dihydro-2,8-dimethyl-1,6-naphthyridine-3-carboxylate | 1050477-44-5 | |
2-cyanoethyl (S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carboxylate | 2640574-73-6 | |
4-(4-Cyano-2-methoxyphenyl)-5-ethoxy-1,4-dihydro-2,8-dimethyl-1,6-naphthyridine-3-carboxylic acid | 1050477-45-6 | |
(S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carboxylic acid | 2640506-74-5 | |
Mavacamten | Isopropylurea | 691-60-1 |
1-Isopropylpyrimidine-2,4,6(1H,3H,5H)-trione | 69998-14-7 | |
6-Chloro-3-isopropylpyrimidine-2,4(1H,3H)-dione | 887581-47-7 | |
Empagliflozin | (3S)-3-[4-[(5-Bromo-2-chlorophenyl)methyl]phenoxy]tetrahydro-furan | 915095-89-5 |
(S)-(2-chloro-5-iodophenyl)(4-((tetrahydrofuran-3-yl)oxy)phenyl)methanone | 915095-87-3 | |
(3S)-3-(4-(2-chloro-5-iodobenzyl)phenoxy)tetrahydrofuran | 915095-94-2 | |
(1S)-1,5-anhydro-2,3,4,6-tetra-O-acteyl-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydrofuran-3-yl]oxy]phenyl] methyl]phenyl]-D-Glucitol | 915095-99-7 | |
Dapagliflozin | (2S,3R,4S,5S,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(hydroxyMethyl) -2-Methoxytetrahydro-2H-pyran-3,4,5-triol | 714269-57-5 |
(1S)-1,5-Anhydro-1-C-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-D-glucitol tetraacetate | 461432-25-7 | |
Canagliflozin | (2S,3R,4S,5S,6R)-2-(3-((5-(4-fluorophenyl)thiophen-2-yl)Methyl)-4-Methylphenyl)-tetrahydro-6-(hydroxyMethyl)-2-Methoxy-2H-pyran-3,4,5-triol | 1358581-37-9 |
(1S)-1,5-Anhydro-1-C-[3-[[5-(4-fluorophenyl)-2-thienyl]methyl]-4-methylphenyl]-D-glucitol tetraacetate | 866607-35-4 | |
Bexagliflozin | 4-Bromo-1-chloro-2-(4-(2-cyclopropoxyethoxy)benzyl)benzene | 1118567-45-5 |
1-Chloro-2-[[4-[2-(cyclopropyloxy)ethoxy]phenyl]methyl]-4-iodobenzene | 1400980-44-0 | |
(2R,3R,4R,5S,6S)-2-(acetoxymethyl)-6-(4-chloro-3-(4-(2-cyclopropoxyethoxy) benzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate | 2251691-23-1 | |
Orforglipron | 1-(Cyanomethyl)-N-methyl-N-phenyl-5-[(4S)-tetrahydro-2,2-dimethyl-2H-pyran-4-yl]-1H-Indole-2-carboxamide | 2212021-80-0 |
1-[(1S,2S)-1-cyano-2-methylcyclopropyl]-N-methyl-N-phenyl-5-[(4S)-tetrahydro-2,2-dimethyl-2H-pyran-4-yl]-1H-Indole-2-carboxamide | 2212021-81-1 | |
(4S)-2-(4-Fluoro-3,5-dimethylphenyl)-3-[3-(4-fluoro-1-methylindazol-5-yl)-2-oxoimidazol-1-yl]-4-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxylic acid tert-butyl ester | 2212022-55-2 | |
1-[(4S)-2-(4-fluoro-3,5-dimethylphenyl)-4,5,6,7-tetrahydro-4-methyl-2H-pyrazolo[4,3-c]pyridin-3-yl]-3-(4-fluoro-1-methyl-1H-indazol-5-yl)-1,3-dihydro-2H-Imidazol-2-one | 2212022-56-3 | |
5-((4S)-2,2-Dimethyloxan-4-yl)-1-[(1S,2S)-2-methyl-1-(5-oxo-4H-1,2,4-oxadiazol-3-yl)cyclopropyl]indole-2-carboxylic acid | 2212021-83-3 | |
Resmetirom | 3,5-Dichloro-4-[[6-chloro-5-(1-methylethyl)-3-pyridazinyl]oxy]benzenamine | 920509-27-9 |
6-(4-Amino-2,6-dichlorophenoxy)-4-(1-methylethyl)-3(2H)-pyridazinone | 920509-28-0 | |
N-Cyanoacetylurethane | 6629-04-5 | |
Ethyl N-[2-cyano-2-[2-[3,5-dichloro-4-[[1,6-dihydro-5-(1-methylethyl)-6-oxo-3-pyridazinyl]oxy]phenyl]hydrazinylidene]acetyl]carbamate | 920509-33-7 | |
Upadacitinib Hemihydrate | (3S,4R)-benzyl 3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl) pyrrolidine-1-carboxylate | 2095311-51-4 |
(3S,4R)-3-ethyl-4-[3-[(4-methylphenyl)sulfonyl]-3H-imidazo[1,2-a]pyrrolo [2,3-e]pyrazin-8-yl]-1-Pyrrolidinecarboxylic acid phenylmethyl ester | 1708997-42-5 | |
8-((3S,4S)-4-ethylpyrrolidin-3-yl)-3-tosyl-3a,9a-dihydro-3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazine | 1428243-28-0 | |
8-[(3R,4S)-4-ethyl-3-pyrrolidinyl]-3H-Imidazo[1,2-a]pyrrolo[2,3-e]pyrazine hydrochloride (1:2) | 2050038-84-9 | |
(3S,4R)-3-ethyl-4-(3-tosyl-3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide | 2411540-30-0 | |
Deucravacitinib | 4,6-Dichloro-N-(methyl-d3)-3-pyridazinecarboxamide | 1609393-89-6 |
3-Pyridazinecarboxylic acid, 6-chloro-4-[[2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl]amino]-, methyl ester | 2720564-44-1 | |
6-chloro-4-[[2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl] amino]-3-Pyridazinecarboxylic acid zinc salt (2:1) | 2245111-17-3 | |
Methyl-d3-amine hydrochloride | 7436-22-8 | |
6-[(cyclopropylcarbonyl)amino]-4-[[2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl]amino]-3-Pyridazinecarboxylic acid zinc salt (2:1) | 2245111-19-5 | |
Baricitinib | 1-(ethylsulfonyl)-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]-3-Azetidineacetonitrile | 1919837-50-5 |
4-[1-[3-(cyanomethyl)-1-(ethylsulfonyl)-3-azetidinyl]-1H-pyrazol-4-yl]-7H-Pyrrolo[2,3-d]pyrimidine-7-carboxylic acid 1,1-dimethylethyl ester | 2055723-13-0 | |
Iptacopan | tert-Butyl 4-formyl-5-methoxy-7-methyl-indole-1-carboxylate | 1481631-51-9 |
tert-Butyl 4-(((2S,4S)-4-ethoxy-2-(4-(methoxycarbonyl)phenyl)piperidin-1-yl)methyl)-5-methoxy-7-methyl-1H-indole-1-carboxylate | 2361158-02-1 | |
Fezolinetant | (R)-3-methyl-5-(8-methyl-7-tosyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)-1,2,4-thiadiazole | / |
(8R)-5,6,7,8-Tetrahydro-8-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1,2,4-triazolo[4,3-a]pyrazine | 1429558-08-6 | |
Roxadustat | 4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid methyl ester | 1421312-34-6 |
4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid ethyl ester | 1809286-36-9 | |
4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid | 1421312-35-7 | |
Methyl 2-(4-hydroxy-1-methyl-7-phenoxyisoquinoline-3-carboxamido) acetate | 1421312-36-8 | |
Elagolix Sodium | 3-[(R)-2-(tert-Butoxycarbonyl)amino-2-phenylethyl]-5-(2-fluoro-3-methoxyphenyl)-1-(2-fluoro-6-trifluoromethylbenzyl)-6-methyl-1H-pyrimidine-2,4-dione | 830346-51-5 |
3-[(2R)-2-Amino-2-phenylethyl]-5-(2-fluoro-3-methoxyphenyl)-1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methyl-2,4(1H,3H)-pyrimidinedione | 830346-50-4 | |
Ethyl (R)-4-((2-(5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-(trifluoromethyl)benzyl)-4-methyl-2,6-dioxo-3,6-dihydropyrimidin-1(2H)-yl)-1-phenylethyl)amino)butanoate Hydrochloride | 1150560-46-5 | |
Acalabrutinib | N-Pyridin-2-yl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzamide | 1383385-64-5 |
[4-[(Pyridin-2-yl)carbamoyl]phenyl]boronic acid | 850568-25-1 | |
4-[8-amino-3-(2S)-2-pyrrolidinylimidazo[1,5-a]pyrazin-1-yl]-N-2-pyridinyl-Benzamide | 1420478-90-5 | |
Abemaciclib | 6-Bromo-4-fluoro-1-isopropyl-2-methyl-1H-benzo[d]imidazole | 1231930-33-8 |
4-fluoro-1-isopropyl-2-Methyl-6-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan -2-yl)-1H-benzo[d]iMidazole | 1231930-37-2 | |
6-(2-chloro-5-fluoro-4-pyriMidinyl)-4-fluoro-2-Methyl-1-(1-Methylethyl)-1H-BenziMidazole | 1231930-42-9 | |
5-((4-Ethylpiperazin-1-yl)methyl)pyridin-2-amine | 1180132-17-5 | |
Apalutamide | 1-((3-fluoro-4-(methylcarbamoyl)phenyl)amino)cyclobutanecarboxylic acid | 2227589-22-0 |
methyl 1-((3-fluoro-4-(methylcarbamoyl)phenyl)amino)cyclobutanecarboxylate | 2227589-23-1 | |
5-Amino-3-(trifluoromethyl)-2-pyridinecarbonitrile | 573762-62-6 | |
Enzalutamide | 4-Bromo-2-fluoro-N-methylbenzamide | 749927-69-3 |
4-Amino-2-Fluoro-N-Methylbenzamide | 915087-25-1 | |
N-[3-Fluoro-4-[(methylamino)carbonyl]phenyl]-2-methylalanine | 1289942-66-0 | |
N-[3-Fluoro-4-[(methylamino)carbonyl]phenyl]-2-methylalanine methyl ester | 1332524-01-2 | |
Alectinib Hydrochloride | 6-Cyano-2-[1-[4-ethyl-3-[4-(4-morpholinyl)-1-piperidinyl]phenyl]-1-methylethyl]-1H-indole-3-carboxylic acid 1,1-dimethylethyl ester hydrochloride | 1256584-77-6 |
6-Cyano-2-[1-[4-ethyl-3-[4-(4-morpholinyl)-1-piperidinyl]phenyl]-1-methylethyl]-1H-Indole-3-carboxylic acid | 1256584-78-7 | |
Pirtobrutinib | 5-amino-3-[4-(aminomethyl)phenyl]-1-[(1S)-2,2,2-trifluoro-1-methylethyl]-1H-Pyrazole-4-carboxamide | 2764851-20-7 |
5-Fluoro-2-methoxybenzoyl chloride | 704-03-0 | |
N-[[4-[5-Amino-4-cyano-1-[(1S)-2,2,2-trifluoro-1-methylethyl]-1H-pyrazol-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide | 2642629-21-6 | |
Eltrombopag olamine | 3-bromo-2-methoxyaniline | 116557-46-1 |
3''-Amino-2''-Hydroxy-Biphenyl-3-Carboxylic Acid | 376592-93-7 | |
2-(3,4-Dimethylphenyl)-1,2-Dihydro-5-Methyl-3h-Pyrazol-3-One | 277299-70-4 | |
1-(3,4-Dimethylphenyl)-3-Methyl-3-Pyrazolin-5-One | 18048-64-1 | |
Parecoxib | 5-Methyl-3,4-Diphenylisoxazole | 37928-17-9 |
Cangrelor | (2r,3s,4r,5r)-2-(Hydroxymethyl)-5-(6-((2-(Methylthio)Ethyl)Amino)-2-((3,3,3-Trifluoropropyl)Thio)-9h-Purin-9-Yl)Tetrahydrofuran-3,4-Diol | 163706-58-9 |
Phosphonic Acid, P,P'-(Dichloromethylene)Bis-, Compd. With N,N-Dibutyl-1-Butanamine (1:1) | 163706-61-4 | |
Ruxolitinib | (R)-3-(4-Bromo-1h-Pyrazol-1-Yl)-3-Cyclopentylpropanenitrile | 1146629-83-5 |
(R)-3-Cyclopentyl-3-(4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)-1h-Pyrazol-1-Yl)Propanenitrile | 1146629-84-6 | |
3-Cyclopentylacrylonitrile | 591769-05-0 | |
Rimegepant | 2-Oxo-1-(4-Piperidinyl)-2,3-Dihydro-1h-Imidazo[4,5-B]Pyridine Dihydrochloride | 781649-84-1 |
(R)-9-((Triisopropylsilyl)Oxy)-6,7,8,9-Tetrahydro-5h-Cyclohepta[B]Pyridin-5-Onehydrochloride | 1190363-45-1 | |
(5s,6s,9r)-6-(2,3-Difluorophenyl)-9-((Triisopropylsilyl)Oxy)-6,7,8,9-Tetrahydro-5h-Cyclohepta[B]Pyridin-5-Aminedihydrochloride | 1373116-04-1 | |
1-(1-(1h-Imidazole-1-Carbonyl)Piperidin-4-Yl)-1h-Imidazo[4,5-B]Pyridin-2(3h)-One | 1373116-06-3 | |
Ubrogepant | (S)-2'-Oxo-1',2',5,7-Tetrahydrospiro[Cyclopenta[B]Pyridine-6,3'-Pyrrolo[2,3-B]Pyridine]-3-Carboxylic Acid | 1375541-21-1 |
(3s,5s,6r)-6-Methyl-2-Oxo-5-Phenyl-1-(2,2,2-Trifluoroethyl)Piperidine-3-Aminium 4-Nitrobenzoate | 1456803-37-4 |