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Final API

Chemical Name

Cas no

Sacubitril Valsartan
(LCZ696)

(R,E)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)aMino)-2-Methylpent -2-enoic acid

1012341-48-8


(2R,4S)-5-(Biphenyl-4-yl)-4-[(tert-butoxycarbonyl)amino]-2-methylpentanoic acid

1012341-50-2


(2R,4S)-4-Amino-5-(biphenyl-4-yl)-2-methylpentanoic acid ethyl ester hydrochloride

149690-12-0


Sacubitril Calcium

1369773-39-6


Sacubitril Sodium

149690-05-1

Finerenone 

2-Cyanoethyl 4-(4-cyano-2-methoxyphenyl)-1,4,5,6-tetrahydro-2,8-dimethyl-5-oxo-1,6-naphthyridine-3-carboxylate

1050477-43-4


2-Cyanoethyl 4-(4-cyano-2-methoxyphenyl)-5-ethoxy-1,4-dihydro-2,8-dimethyl-1,6-naphthyridine-3-carboxylate

1050477-44-5


2-cyanoethyl (S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carboxylate

2640574-73-6


4-(4-Cyano-2-methoxyphenyl)-5-ethoxy-1,4-dihydro-2,8-dimethyl-1,6-naphthyridine-3-carboxylic acid

1050477-45-6


(S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carboxylic acid

2640506-74-5

Mavacamten

Isopropylurea

691-60-1


1-Isopropylpyrimidine-2,4,6(1H,3H,5H)-trione

69998-14-7


6-Chloro-3-isopropylpyrimidine-2,4(1H,3H)-dione

887581-47-7

Empagliflozin

(3S)-3-[4-[(5-Bromo-2-chlorophenyl)methyl]phenoxy]tetrahydro-furan

915095-89-5


(S)-(2-chloro-5-iodophenyl)(4-((tetrahydrofuran-3-yl)oxy)phenyl)methanone

915095-87-3


(3S)-3-(4-(2-chloro-5-iodobenzyl)phenoxy)tetrahydrofuran

915095-94-2


(1S)-1,5-anhydro-2,3,4,6-tetra-O-acteyl-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydrofuran-3-yl]oxy]phenyl] methyl]phenyl]-D-Glucitol

915095-99-7

Dapagliflozin

(2S,3R,4S,5S,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(hydroxyMethyl) -2-Methoxytetrahydro-2H-pyran-3,4,5-triol

714269-57-5


(1S)-1,5-Anhydro-1-C-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-D-glucitol tetraacetate

461432-25-7

Canagliflozin 

(2S,3R,4S,5S,6R)-2-(3-((5-(4-fluorophenyl)thiophen-2-yl)Methyl)-4-Methylphenyl)-tetrahydro-6-(hydroxyMethyl)-2-Methoxy-2H-pyran-3,4,5-triol

1358581-37-9


(1S)-1,5-Anhydro-1-C-[3-[[5-(4-fluorophenyl)-2-thienyl]methyl]-4-methylphenyl]-D-glucitol tetraacetate

866607-35-4

Bexagliflozin

4-Bromo-1-chloro-2-(4-(2-cyclopropoxyethoxy)benzyl)benzene

1118567-45-5


1-Chloro-2-[[4-[2-(cyclopropyloxy)ethoxy]phenyl]methyl]-4-iodobenzene

1400980-44-0


(2R,3R,4R,5S,6S)-2-(acetoxymethyl)-6-(4-chloro-3-(4-(2-cyclopropoxyethoxy) benzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate

2251691-23-1

Orforglipron

1-(Cyanomethyl)-N-methyl-N-phenyl-5-[(4S)-tetrahydro-2,2-dimethyl-2H-pyran-4-yl]-1H-Indole-2-carboxamide

2212021-80-0


1-[(1S,2S)-1-cyano-2-methylcyclopropyl]-N-methyl-N-phenyl-5-[(4S)-tetrahydro-2,2-dimethyl-2H-pyran-4-yl]-1H-Indole-2-carboxamide

2212021-81-1


(4S)-2-(4-Fluoro-3,5-dimethylphenyl)-3-[3-(4-fluoro-1-methylindazol-5-yl)-2-oxoimidazol-1-yl]-4-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxylic acid tert-butyl ester

2212022-55-2


1-[(4S)-2-(4-fluoro-3,5-dimethylphenyl)-4,5,6,7-tetrahydro-4-methyl-2H-pyrazolo[4,3-c]pyridin-3-yl]-3-(4-fluoro-1-methyl-1H-indazol-5-yl)-1,3-dihydro-2H-Imidazol-2-one

2212022-56-3


5-((4S)-2,2-Dimethyloxan-4-yl)-1-[(1S,2S)-2-methyl-1-(5-oxo-4H-1,2,4-oxadiazol-3-yl)cyclopropyl]indole-2-carboxylic acid

2212021-83-3

Resmetirom

3,5-Dichloro-4-[[6-chloro-5-(1-methylethyl)-3-pyridazinyl]oxy]benzenamine

920509-27-9


6-(4-Amino-2,6-dichlorophenoxy)-4-(1-methylethyl)-3(2H)-pyridazinone

920509-28-0


N-Cyanoacetylurethane

6629-04-5


Ethyl N-[2-cyano-2-[2-[3,5-dichloro-4-[[1,6-dihydro-5-(1-methylethyl)-6-oxo-3-pyridazinyl]oxy]phenyl]hydrazinylidene]acetyl]carbamate

920509-33-7

Upadacitinib Hemihydrate

(3S,4R)-benzyl 3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl) pyrrolidine-1-carboxylate

2095311-51-4


(3S,4R)-3-ethyl-4-[3-[(4-methylphenyl)sulfonyl]-3H-imidazo[1,2-a]pyrrolo [2,3-e]pyrazin-8-yl]-1-Pyrrolidinecarboxylic acid phenylmethyl ester 

1708997-42-5


8-((3S,4S)-4-ethylpyrrolidin-3-yl)-3-tosyl-3a,9a-dihydro-3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazine

1428243-28-0


8-[(3R,4S)-4-ethyl-3-pyrrolidinyl]-3H-Imidazo[1,2-a]pyrrolo[2,3-e]pyrazine hydrochloride (1:2)

2050038-84-9


(3S,4R)-3-ethyl-4-(3-tosyl-3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide

2411540-30-0

Deucravacitinib

4,6-Dichloro-N-(methyl-d3)-3-pyridazinecarboxamide

1609393-89-6


3-Pyridazinecarboxylic acid, 6-chloro-4-[[2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl]amino]-, methyl ester

2720564-44-1


6-chloro-4-[[2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl] amino]-3-Pyridazinecarboxylic acid zinc salt (2:1) 

2245111-17-3


Methyl-d3-amine hydrochloride

7436-22-8


6-[(cyclopropylcarbonyl)amino]-4-[[2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl]amino]-3-Pyridazinecarboxylic acid zinc salt (2:1)

2245111-19-5

Baricitinib

1-(ethylsulfonyl)-3-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl]-3-Azetidineacetonitrile 

1919837-50-5


4-[1-[3-(cyanomethyl)-1-(ethylsulfonyl)-3-azetidinyl]-1H-pyrazol-4-yl]-7H-Pyrrolo[2,3-d]pyrimidine-7-carboxylic acid 1,1-dimethylethyl ester

2055723-13-0

Iptacopan 

tert-Butyl 4-formyl-5-methoxy-7-methyl-indole-1-carboxylate

1481631-51-9


tert-Butyl 4-(((2S,4S)-4-ethoxy-2-(4-(methoxycarbonyl)phenyl)piperidin-1-yl)methyl)-5-methoxy-7-methyl-1H-indole-1-carboxylate

2361158-02-1

Fezolinetant

(R)-3-methyl-5-(8-methyl-7-tosyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazin-3-yl)-1,2,4-thiadiazole

/


(8R)-5,6,7,8-Tetrahydro-8-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1,2,4-triazolo[4,3-a]pyrazine

1429558-08-6

Roxadustat

4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid methyl ester

1421312-34-6


4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid ethyl ester

1809286-36-9


4-Hydroxy-1-methyl-7-phenoxy-3-isoquinolinecarboxylic acid

1421312-35-7


Methyl 2-(4-hydroxy-1-methyl-7-phenoxyisoquinoline-3-carboxamido) acetate

1421312-36-8

Elagolix Sodium

3-[(R)-2-(tert-Butoxycarbonyl)amino-2-phenylethyl]-5-(2-fluoro-3-methoxyphenyl)-1-(2-fluoro-6-trifluoromethylbenzyl)-6-methyl-1H-pyrimidine-2,4-dione

830346-51-5


3-[(2R)-2-Amino-2-phenylethyl]-5-(2-fluoro-3-methoxyphenyl)-1-[[2-fluoro-6-(trifluoromethyl)phenyl]methyl]-6-methyl-2,4(1H,3H)-pyrimidinedione

830346-50-4


Ethyl (R)-4-((2-(5-(2-fluoro-3-methoxyphenyl)-3-(2-fluoro-6-(trifluoromethyl)benzyl)-4-methyl-2,6-dioxo-3,6-dihydropyrimidin-1(2H)-yl)-1-phenylethyl)amino)butanoate Hydrochloride

1150560-46-5

Acalabrutinib

N-Pyridin-2-yl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzamide

1383385-64-5


[4-[(Pyridin-2-yl)carbamoyl]phenyl]boronic acid

850568-25-1


4-[8-amino-3-(2S)-2-pyrrolidinylimidazo[1,5-a]pyrazin-1-yl]-N-2-pyridinyl-Benzamide

1420478-90-5

Abemaciclib

6-Bromo-4-fluoro-1-isopropyl-2-methyl-1H-benzo[d]imidazole

1231930-33-8


4-fluoro-1-isopropyl-2-Methyl-6-(4,4,5,5-tetraMethyl-1,3,2-dioxaborolan -2-yl)-1H-benzo[d]iMidazole

1231930-37-2


6-(2-chloro-5-fluoro-4-pyriMidinyl)-4-fluoro-2-Methyl-1-(1-Methylethyl)-1H-BenziMidazole

1231930-42-9


5-((4-Ethylpiperazin-1-yl)methyl)pyridin-2-amine

1180132-17-5

Apalutamide

1-((3-fluoro-4-(methylcarbamoyl)phenyl)amino)cyclobutanecarboxylic acid

2227589-22-0


methyl 1-((3-fluoro-4-(methylcarbamoyl)phenyl)amino)cyclobutanecarboxylate

2227589-23-1


5-Amino-3-(trifluoromethyl)-2-pyridinecarbonitrile

573762-62-6

Enzalutamide

4-Bromo-2-fluoro-N-methylbenzamide

749927-69-3


4-Amino-2-Fluoro-N-Methylbenzamide

915087-25-1


N-[3-Fluoro-4-[(methylamino)carbonyl]phenyl]-2-methylalanine

1289942-66-0


N-[3-Fluoro-4-[(methylamino)carbonyl]phenyl]-2-methylalanine methyl ester

1332524-01-2

Alectinib Hydrochloride

6-Cyano-2-[1-[4-ethyl-3-[4-(4-morpholinyl)-1-piperidinyl]phenyl]-1-methylethyl]-1H-indole-3-carboxylic acid 1,1-dimethylethyl ester hydrochloride

1256584-77-6


6-Cyano-2-[1-[4-ethyl-3-[4-(4-morpholinyl)-1-piperidinyl]phenyl]-1-methylethyl]-1H-Indole-3-carboxylic acid

1256584-78-7

Pirtobrutinib 

5-amino-3-[4-(aminomethyl)phenyl]-1-[(1S)-2,2,2-trifluoro-1-methylethyl]-1H-Pyrazole-4-carboxamide

2764851-20-7


5-Fluoro-2-methoxybenzoyl chloride

704-03-0


N-[[4-[5-Amino-4-cyano-1-[(1S)-2,2,2-trifluoro-1-methylethyl]-1H-pyrazol-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide

2642629-21-6

Eltrombopag olamine

3-bromo-2-methoxyaniline

116557-46-1


3''-Amino-2''-Hydroxy-Biphenyl-3-Carboxylic Acid

376592-93-7


2-(3,4-Dimethylphenyl)-1,2-Dihydro-5-Methyl-3h-Pyrazol-3-One

277299-70-4


1-(3,4-Dimethylphenyl)-3-Methyl-3-Pyrazolin-5-One

18048-64-1

Parecoxib

5-Methyl-3,4-Diphenylisoxazole

37928-17-9

Cangrelor

(2r,3s,4r,5r)-2-(Hydroxymethyl)-5-(6-((2-(Methylthio)Ethyl)Amino)-2-((3,3,3-Trifluoropropyl)Thio)-9h-Purin-9-Yl)Tetrahydrofuran-3,4-Diol

163706-58-9


Phosphonic Acid, P,P'-(Dichloromethylene)Bis-, Compd. With N,N-Dibutyl-1-Butanamine (1:1)

163706-61-4

Ruxolitinib 

(R)-3-(4-Bromo-1h-Pyrazol-1-Yl)-3-Cyclopentylpropanenitrile

1146629-83-5


(R)-3-Cyclopentyl-3-(4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)-1h-Pyrazol-1-Yl)Propanenitrile

1146629-84-6


3-Cyclopentylacrylonitrile

591769-05-0

Rimegepant

2-Oxo-1-(4-Piperidinyl)-2,3-Dihydro-1h-Imidazo[4,5-B]Pyridine Dihydrochloride

781649-84-1


(R)-9-((Triisopropylsilyl)Oxy)-6,7,8,9-Tetrahydro-5h-Cyclohepta[B]Pyridin-5-Onehydrochloride

1190363-45-1


(5s,6s,9r)-6-(2,3-Difluorophenyl)-9-((Triisopropylsilyl)Oxy)-6,7,8,9-Tetrahydro-5h-Cyclohepta[B]Pyridin-5-Aminedihydrochloride

1373116-04-1


1-(1-(1h-Imidazole-1-Carbonyl)Piperidin-4-Yl)-1h-Imidazo[4,5-B]Pyridin-2(3h)-One

1373116-06-3

Ubrogepant

(S)-2'-Oxo-1',2',5,7-Tetrahydrospiro[Cyclopenta[B]Pyridine-6,3'-Pyrrolo[2,3-B]Pyridine]-3-Carboxylic Acid

1375541-21-1


(3s,5s,6r)-6-Methyl-2-Oxo-5-Phenyl-1-(2,2,2-Trifluoroethyl)Piperidine-3-Aminium 4-Nitrobenzoate

1456803-37-4

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